Formulation and characterization of nanofibers and films with carvedilol prepared by electrospinning and solution casting method

Published in European Journal of Pharmaceutical Sciences, vol. 101, pp. 160–166 (2017) · Elsevier
DOI: 10.1016/j.ejps.2017.02.006

Summary

Carvedilol is a poorly water-soluble cardiovascular drug whose slow dissolution limits its absorption. This study formulates carvedilol together with the water-soluble polymer poly(ethylene oxide) (PEO) into two dosage forms — solvent-cast films and electrospun nanofibres — using water or ethanol/water as benign solvents, and compares them. Infrared spectroscopy confirmed no chemical interaction between the drug and PEO, while differential scanning calorimetry showed the carvedilol had dissolved into the polymer and altered its crystallinity, i.e. it was dispersed rather than present as separate crystals. Both formats released carvedilol faster than the pure drug, and the release rate differed markedly between the cast films and the electrospun fibres — highlighting electrospinning as a way to tune and accelerate the dissolution of poorly soluble drugs.

Authors & Affiliations

Topics

Drug Delivery Dissolution Enhancement Solid Dispersions Oral Films

Materials

Carvedilol Poly(ethylene oxide) (PEO)

Linari Electrospinning Systems

Electrospinning machines by Linari Nanotech
Linari Nanotech designs and manufactures electrospinning systems for nanofiber research and production — including drug-loaded fibres for fast-dissolving dosage forms.
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