Formulation and evaluation of chitosan/polyethylene oxide nanofibers loaded with metronidazole for local infections

Published in European Journal of Pharmaceutical Sciences, vol. 95, pp. 152–160 (2016) · Elsevier
DOI: 10.1016/j.ejps.2016.10.030

Summary

Combining nanofibers with an antimicrobial is a powerful approach for treating local infections, because the fibrous mat can stick to and stay at the site of application while releasing the drug. This study develops biocompatible, biodegradable chitosan/poly(ethylene oxide) (PEO) nanofibers loaded with the antimicrobial metronidazole, produced by environmentally friendly electrospinning of aqueous polymer solutions. Chitosan contributes antibacterial action, biodegradability, and strong bioadhesion — favouring retention at the target site — while PEO enables spinnability. A key point the authors raise is that local infection sites offer only a small fluid volume for drug release, unlike standard pharmacopoeial dissolution tests with large receptor volumes; they therefore argue for release-testing methods that better mimic in-vivo conditions. The nanofibers are characterised for their morphology, drug loading and release behaviour, showing high potential as a bioadhesive local delivery platform.

Authors & Affiliations

Topics

Antimicrobial Nanofibers Local Drug Delivery Bioadhesive Systems Aqueous Electrospinning

Materials

Chitosan Poly(ethylene oxide) (PEO) Metronidazole

Linari Electrospinning Systems

Electrospinning machines by Linari Nanotech
Linari Nanotech designs and manufactures electrospinning systems for nanofiber research and production — including bioadhesive antimicrobial nanofibres for local drug delivery.
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